Neosaxitoxin as a Local Anesthetic | 水產百科網
由AJRodriguez-Navarro著作·2007·被引用63次—Neosaxitoxinisaphycotoxinthatreversiblyblocksthevoltage-gatedsodiumchannelsattheneuronallevel.Itsactivityresultsinblockingtheaxonalconduction, ...
VOLTAGE-GATED sodium channels are responsible for the rising phase of the action potential in the membranes of neurons and most electrically excitable cells.1At least nine distinct voltage-gated sodium channels have been cloned from mammals, being broadly divided by its affinity to tetrodotoxin. NaV1.1, NaV1.2, NaV1.3, and NaV1.7 are highly tetrodotoxin-sensitive, whereas NaV1.5, NaV1.8, and NaV1.9 are tetrodotoxin-resistant to varying degrees.2Many of these channels have specific tissue distributions, determining distinct excitation properties.3
Local anesthetics are compounds that reversibly block the neural conduction by occupying enough sodium channels within an axon to interrupt activity, stopping the depolarization, thus preventing the propagation of action potential and neuronal communication.4
Clinically used local anesthetics such as aminoamides (e.g. ,...
Berde Lab | 水產百科網
Neosaxitoxin | 水產百科網
Neosaxitoxin | 水產百科網
Neosaxitoxin as a Local Anesthetic | 水產百科網
Neosaxitoxin as a local anesthetic | 水產百科網
Neosaxitoxin in Rat Sciatic Block | 水產百科網
Neosaxitoxin versus Traditional Local Anesthetics ... | 水產百科網
Neosaxitoxin | 水產百科網
Neosaxitoxin | 水產百科網
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