Neosaxitoxin in Rat Sciatic Block | 水產百科網
由JSTemplin著作·2015·被引用17次—NeosaxitoxininRatSciaticBlock:ImprovedTherapeuticIndexUsingCombinationswithBupivacaine,withandwithoutEpinephrine.Anesthesiology.2015Oct ...
Background: Neosaxitoxin (NeoSTX) is a site-1 sodium channel blocker undergoing clinical trials as a prolonged-duration local anesthetic. Rat sciatic block and intravenous infusion models were used to assess efficacy and local and systemic toxicities for NeoSTX in saline (NeoSTX-Saline), bupivacaine (Bup), and their combination (NeoSTX-Bup). Exploratory studies evaluated the effects of addition of epinephrine to NeoSTX-Bup (NeoSTX-Bup-Epi).
Methods: Rats received percutaneous sciatic blocks with escalating doses of NeoSTX-Saline or NeoSTX-Bup. Sensory-nocifensive block was assessed using modified hotplate and Von Frey filaments. Motor-proprioceptive function was assessed by extensor postural thrust. Nerves were examined histologically after 7 days and scored on the Estebe-Myers scale. Median lethal dose was estimated for NeoSTX-Saline and in combinations. Accidental intravenous overdose was simulate...
Berde Lab | 水產百科網
Neosaxitoxin | 水產百科網
Neosaxitoxin | 水產百科網
Neosaxitoxin as a Local Anesthetic | 水產百科網
Neosaxitoxin as a local anesthetic | 水產百科網
Neosaxitoxin in Rat Sciatic Block | 水產百科網
Neosaxitoxin versus Traditional Local Anesthetics ... | 水產百科網
Neosaxitoxin | 水產百科網
Neosaxitoxin | 水產百科網
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